- 商品介绍
- 规格参数
- 包装参数
Application
Enzastaurin has been used in splicing analysis to study its effects on splicing of a mutated exon.
Biochem/physiol Actions
It is an orally administered drug. It can induce apoptosis, inhibit angiogenesis and proliferation of cells. Enzastaurin can be used for the treatment of haematological cancers.
Enzastaurin is a potent and PKCβ preferring inhibitor. Also, Enzastaurin inhibits AKT and GSK3β. Enzastaurin acts as anti-angiogenic and antineoplastic agent.
Enzastaurin is a potent and PKCβ proffering inhibitor.
Features and Benefits
This compound is featured on the GSK-3, PKB/Akt and PKC pages of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.
| Quality Segment | 100 |
| assay | ≥98% (HPLC) |
| form | powder |
| storage condition | desiccated |
| color | , light orange to dark orange-red |
| solubility | DMSO: 10 mg/mL, clear (warmed) |
| storage temp. | −20°C |
| SMILES string | N1C(=O)C(=C(C1=O)c6c7c([n](c6)C)cccc7)c2c3c([n](c2)C4CCN(CC4)Cc5ncccc5)cccc3 |
| InChI | 1S/C32H29N5O2/c1-35-19-25(23-9-2-4-11-27(23)35)29-30(32(39)34-31(29)38)26-20-37(28-12-5-3-10-24(26)28)22-13-16-36(17-14-22)18-21-8-6-7-15-33-21/h2-12,15,19-20,22H,13-14,16-18H2,1H3,(H,34,38,39) |
| InChI key | AXRCEOKUDYDWLF-UHFFFAOYSA-N |
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¥ 1563.36
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¥ 1866.29
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¥ 4173.75
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¥ 2883.61
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