- 商品介绍
- 规格参数
- 包装参数
General description
Apratastat is one of the thiomorpholine sulfonamide hydroxymate selective inhibitors of ADAM17 (a disintegrin and metalloproteinase).
Biochem/physiol Actions
Apratastat (TMI-005) is an orally active, potent and selective dual inhibitor of disintegrin metalloenzyme 17 (ADAM17/ TACE) and matrix metalloprotease (MMP).
Apratastat is an orally active, potent and selective dual inhibitor of disintegrin metalloenzyme 17 (ADAM17/ TACE) and matrix metalloprotease (MMP).
| Quality Segment | 100 |
| assay | ≥98% (HPLC) |
| form | powder |
| color | white to beige |
| solubility | DMSO: 20 mg/mL, clear |
| storage temp. | 2-8°C |
| SMILES string | O=S(N1CCSC(C)(C)[C@@H]1C(NO)=O)(C2=CC=C(OCC#CCO)C=C2)=O |
| InChI | 1S/C17H22N2O6S2/c1-17(2)15(16(21)18-22)19(9-12-26-17)27(23,24)14-7-5-13(6-8-14)25-11-4-3-10-20/h5-8,15,20,22H,9-12H2,1-2H3,(H,18,21)/t15-/m0/s1 |
| InChI key | MAVDNGWEBZTACC-HNNXBMFYSA-N |
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| 重量(kg) |
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询价
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¥ 805.47
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¥ 3683.17
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¥ 3895.14
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¥ 2290.18
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¥ 4110.85
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¥ 907.59
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¥ 1334.26
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¥ 1327.84
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¥ 1047.15
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询价
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¥ 1540.85
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¥ 2024.55
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¥ 1164.64
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