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General description
一种跨膜Ca2+通量阻滞剂（IC50 = 7 µM），可减弱辣椒素诱导的阳离子通道开放。抑制从对兰尼碱敏感的细胞内Ca2+贮藏中，Ca2+-诱导的Ca2+释放。抑制K+-刺激的儿茶酚胺分泌(IC50 = 6 µM)。
Biochem/physiol Actions
主靶
跨膜Ca2+通量的阻断剂
产物不与ATP竞争。
可逆：否
细胞可渗透性：否
靶标IC50：7 µM阻断跨膜Ca2+通量；6 µM抑制K+-刺激的儿茶酚胺分泌
Other Notes
Merck Index 13, 8379.
Phillippe, M. and Basa, A. 1996.Biochem.Biophys.Res. Commun.221, 656.
Buratti, R., et al. 1995.Biochem.Biophys.Res. Commun.213, 1082.
Hamilton, M.G. and Lundy, P.M. 1995.J. Pharmacol.Exp.Ther.273, 940.
Gomis, A., et al. 1994.Biochem.Pharmacol.47, 225.
Stjame, P., et al. 1994.Acta Otolaryngol.114, 651.
Ma, J. 1993.J. Gen.Physiol.102, 1031.
Legal Information
CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany
Disclaimer
毒性：有害（C）
| Quality Level | 100 |
| description | Merck USA index - 14, 8300 |
| form | solid |
| manufacturer/tradename | Calbiochem® |
| storage condition | OK to freeze,desiccated |
| color | red-black |
| solubility | ammonia: soluble,water: soluble |
| shipped in | ambient |
| storage temp. | 10-30°C |
| 长度(mm) | |
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