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Biochem/physiol Actions
BMS-470539 is a highly potent and selective melanocortin-1 receptor (MC-1R; MC1R) agonist (AMP stimulation EC50 = 11.6/16.2/16.8 nM using B16/HBL/CHO-MC1R; little or no potency toward MC2R, MC3R MC4R MC5R) with anti-inflammatory efficacy in mice in vivo (15-100 μmol/kg via i.v. or s.c. 0.5-1 h prior to 1 μg LPS s.c.).
Highly potent and selective melanocortin-1 receptor (MC-1R; MC1R) agonist with anti-inflammatory efficacy in mice in vivo.
Disclaimer
Hygroscopic
| Quality Level | 100 |
| assay | ≥98% (HPLC) |
| form | powder |
| storage condition | desiccated |
| color | white to beige |
| solubility | H2O: 2 mg/mL, clear (Warmed) |
| storage temp. | -10 to -25°C |
| SMILES string | CCCC(C1(C2=CC=CC=C2)CCN(CC1)C([C@H](NC([C@@H](N)CC3=CN=CN3C)=O)CC4=CC=C(C=C4)OC)=O)=O.[2HCl] |
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¥ 2528.88
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¥ 1683.78
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¥ 9207.92
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¥ 4173.75
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¥ 2883.61
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¥ 4390.38
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¥ 3812.28
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¥ 2573.97
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¥ 2666.57
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¥ 954.17
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¥ 8072.66
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